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T12404 |
CCK-A receptor inhibitor 1
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cholecystokinin
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T13261 |
CCK-B Receptor Antagonist 1
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Others
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CCK-B Receptor Antagonist 1 is a cholecystokinin B (CCK-B) receptor agonist and has the potential of reducing the secretion of gastric acid. |
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T10707 |
CCK-B Receptor Antagonist 2
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Others
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CCK-B Receptor Antagonist 2 is a potent and orally active antagonist of Gastrin/CCK-B (IC50: 0.43 nM). It also inhibits gastrin/CCK-A activity (IC50: 1.82 μM). |
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TP1197 |
Sincalide
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SQ19844,CCK-8,Cholecystokinin octapeptide |
Others
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Sincalide (CCK-8) is a cholecystokinetic drug administered by injection to aid in diagnosing disorders of the gallbladder and pancreas. It is the 8-amino acid C-terminal fragment of cholecystokinin. |
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T1052 |
Proglumide
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cholecystokinin
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Proglumide (Binoside) is a cholecystokinin antagonist, which blocks both the CCKA and CCKB subtypes. Proglumide is a drug that exerts an inhibitory effect on gastric secretion and reduces gastrointestinal motility. It is... |
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TQ0062 |
Nastorazepide
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Z-360 |
cholecystokinin
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Nastorazepide (Z-360) is a selective, orally available antagonist of gastrin/cholecystokinin 2 (CCK-2) receptor with potential antineoplastic activity. |
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T2312 |
Loxiglumide
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CR-1505 |
cholecystokinin
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Loxiglumide (CR-1505) is an antagonist of cholecystokinin (CCK-1) receptor. |
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T4579 |
Pentagastrin
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ICI-50123 |
Others
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cholecystokinin
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Pentagastrin (ICI-50123) is a synthetic polypeptide that has effects like gastrin when given parenterally, which can cause the secretion and synthesis of salivary proteins. |
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T14932 |
Ceruletide
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Cerulein,Caerulein,FI-6934 |
cholecystokinin
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Ceruletide (Caerulein) is a potent agonist of cholecystokinin receptor and it also is a safe and effective cholecystokinetic agent. It has a direct spasmogenic effect on the gallbladder muscle and bile ducts. |
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T9343 |
N-Cbz-DL-tryptophan
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cholecystokinin
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N-Cbz-DL-tryptophan is a cholecystokinin receptor antagonist, abolished the response of the isolated heart to CCK-8. |
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T14932L |
Ceruletide Ammonium acetate
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FI-6934 Ammonium acetate,Caerulein Ammonium acetate,Ceruletide Ammonium acetate (17650-98-5 free base) |
cholecystokinin
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Ceruletide Ammonium acetate (FI-6934 Ammonium acetate) is a cholecystokinin (CCK) receptor agonist. Ceruletide Ammonium acetate is a safe and effective cholecystokinetic agent and small bowel and exocrine pancreatic stim... |
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TP1931L1 |
[D-Arg1,D-Phe5,D-Trp7,9,Leu11]-Substance P acetate
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[D-Arg1,D-Phe5,D-Trp7,9,Leu11]-Substance P acetate(96736-12-8 free base) |
cholecystokinin
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[D-Arg1,D-Phe5,D-Trp7,9,Leu11]-Substance P acetate ([D-Arg1,D-Phe5,D-Trp7,9,Leu11]-Substance P acetate (96736-12-8 free base)) is a broad spectrum neuropeptide inverse agonist and antagonist. Potent full inverse agonist ... |
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T15101 |
Devazepide
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L-364,718,MK-329 |
Others
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Devazepide is a competitive and orally active nonpeptide antagonist of cholecystokinin (CCK) receptor (IC50s: 81 pM, 45 pM, and 245 nM for rat pancreatic, bovine gallbladder and guinea pig brain CCK receptors, respective... |
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T28340 |
PD-135666
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PD 135666 |
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PD-135666 is an antagonist of CCK receptor. |
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T26483 |
A-65186
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A65186 |
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A 65186 is a Type A Cholecystokinin (CCK) receptor antagonist. |
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T23886 |
Cholecystokinin (27-32)-amide
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Cholecystokinin (27-32)-NH2 |
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Cholecystokinin (27-32)-amide is a CCK receptor antagonist. |
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T22666 |
CI-988
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CI 988 |
Others
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CCK2 (CCK-B) receptor antagonist |
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T13084 |
Tarazepide
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Others
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Tarazepide is a potent and specific antagonist of CCK-A receptor. |
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T27014 |
CI-1015
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CI1015,CI 1015,PD 144598 |
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CI-1015 is a CCK-B receptor antagonist with oral activity. |
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T29502 |
A 70874
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A-70874,A70874 |
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A70874 has high selectivity and potency for cholecystokinin (CCK) a receptor. |
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T25553 |
Jmv 332
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Jmv-332,Jmv332 |
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Jmv 332 is a cyclic analog of the C-terminal hexapeptide of CCK. It is a CCK/gastrin receptor agonist. |
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T27774 |
L-740093
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L 740093 |
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L-740093 is a specific antagonist of CCK-B receptor. |
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T28342 |
PD-149164
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PD 149164,PD149164 |
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PD-149164 is an agonist of the CCK-A receptor. |
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T17274 |
YM022
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CCR
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YM022 is a highly effective and selective gastrin/cholecystokinin (CCK)-B receptor antagonist. YM022 can inhibit gastrin-induced gastric acid secretion and histidine decarboxylase activation in vivo. YM022 shows the Ki v... |
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T27900 |
LY 219057
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LY-219057,LY219057 |
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LY 219057 is a potent, competitive, and specific antagonist of CCK receptor on the exocrine pancreas. |
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T27772 |
L-736380
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L-736,380,L 736380,L736,380,L 736,380 |
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L-736380 is a CCK-B receptor antagonist. L-736,380 dose-dependently inhibited gastric acid secretion in anesthetized rats (ID(50), 0.064 mg/kg) and ex vivo binding of [(125)I]CCK-8S in BKTO mice brain membranes (ED(50), ... |
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T28331 |
PD 136450
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Cam1189,PD136450,Cam-1189,PD-136450,Cam 1189 |
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Cholecystokinin type B receptor antagonist PD-136,450 is a partial secretory agonist in the stomach and a full agonist in the pancreas of the rat. Gastrin (cholecystokinin type B (CCK-B)) receptor antagonists may help to... |
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T62039 |
L-365260 hemihydrate
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L-365260 hemihydrate is a selective, orally active non-peptide gastrin and brain cholecystokinin receptor (CCK-B) antagonist, demonstrating competitive interaction with guinea pig stomach gastrin and brain CCK receptors ... |
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TP1931 |
[D-Arg1,D-Phe5,D-Trp7,9,Leu11]-Substance P
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Broad spectrum neuropeptide inverse agonist and antagonist. Potent full inverse agonist for the ghrelin receptor (EC50 = 5.2 nM); diminishes constitutive ghrelin receptor signaling. Also antagonist at tachykinin, bradyki... |
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T8761 |
[Leu15]-Gastrin I human
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Amino Acid Sequence Glp-Gly-Pro-Trp-Leu-Glu-Glu-Glu-Glu-Glu-Ala-Tyr-Gly-Trp-Leu-Asp-Phe-NH2 |
Others
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[Leu15]-Gastrin I human (Amino Acid Sequence Glp-Gly-Pro-Trp-Leu-Glu-Glu-Glu-Glu-Glu-Ala-Tyr-Gly-Trp-Leu-Asp-Phe-NH2) encodes for the protein [Leu15]-Gastrin I in human. In human chromosome, the gene GAST is localized on... |
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T68482 |
CE-326597
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CE-326597 is a potent and selective CCK1R agonist. The type 1 cholecystokinin receptor (CCK1R) has multiple physiologic roles relating to nutrient homeostasis,including mediation of postcibal satiety. The type 1 cholecy... |
